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Pharmaceutical Intermediates

Full official intermediate catalog + key intermediates with CEP / DMF / GMP / cold-chain qualifications and capacity details · each quotable via RFQ

Featured ProductsProven track record · documents on request

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Dealt

Orforglipron intermediates

样品订单(各 500g)+ 0.5KG 复购

2 deals completed · latest 2026-09-21

Documents in progress

Dealt

PINACOLONE

两用物项贸易品类

2 deals completed · latest 2026-01-19

Documents in progress

Dealt

4-(3-Bromophenyl)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline

CAS 543737-10-6

1 deal completed · latest 2026-07-08

Documents in progress

By Therapeutic Area of Target Drug

Click a class to filter both sections below; classes follow the target API's primary indication

Qualified Key IntermediatesCEP / DMF / GMP / Cold-chain / Capacity / Price-band details

13 items
Product / CASPurity / Impurity profile (redacted)Synthesis route (redacted)CapacityQualificationsPackaging / Cold-chainMOQ / Price bandAction
Lenacapavir INT-1|N-Boc 手性胺酯
CAS 1620056-47-4 · Antivirals
Target drug: lenacapavir
高保密
≥99.0%
单杂 ≤0.10%,总杂 ≤0.50%(脱敏)
手性还原 + Boc 保护(脱敏简述)1,200 kg/yr
US DMF
5 kg / 25 kg 桶(铝箔袋内衬)
1 kg
US$ 2,600-3,800 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-2|4-氯-7-硼酸酯吲唑
CAS 2189684-53-3 · Antivirals
Target drug: lenacapavir
高保密
≥98.5%
有关物质谱见 CDA 资料室
吲唑构建 + Miyaura 硼化(脱敏简述)900 kg/yr
US DMF
1 kg / 5 kg 铝瓶
Cold chain
0.5 kg
US$ 4,200-6,000 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-3|环丙烷并环戊烷吡唑乙酸
CAS 1620056-83-8 · Antivirals
Target drug: lenacapavir
高保密
≥99.0%
手性纯度 ≥99.5% ee(脱敏)
双环构建 + 三氟甲基化(脱敏简述)700 kg/yr
US DMF
1 kg 铝瓶
Cold chain
0.5 kg
US$ 5,800-8,200 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-4|3-甲基-3-(甲磺酰基)-1-丁炔
CAS 2109226-54-0 · Antivirals
Target drug: lenacapavir
CDA 后可看
≥98.0%
单杂 ≤0.20%(脱敏)
炔基化 + 砜基引入(脱敏简述)2,400 kg/yr
25 kg 桶
5 kg
US$ 780-1,150 / kg
Unibest Taizhou GMP-like Site
Lenacapavir (GS-6207) API
CAS 2189684-44-2 · Antivirals
Target drug: lenacapavir
高保密
≥99.5%
单杂 ≤0.10%,总杂 ≤0.30%(脱敏)
汇聚式偶联 + 成盐(脱敏简述)300 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶(密闭系统)
Cold chain
100 g
🔒 CDA 后开放
Unibest Nantong cGMP Site
Doravirine INT-1|3-氯-5-[(吡啶基)氧基]苯甲腈
CAS 1155846-86-8 · Antivirals
Target drug: doravirine
CDA 后可看
≥99.0%
单杂 ≤0.15%(脱敏)
芳香亲核取代成醚(脱敏简述)3,600 kg/yr
US DMFEU GMP
25 kg 桶
10 kg
US$ 420-620 / kg
Qualified Partner — East China API Works
Doravirine INT-2|3-氯-5-碘苯酚
CAS 861347-86-6 · Antivirals
Target drug: doravirine
≥99.0%
单杂 ≤0.15%(脱敏)
选择性碘代(脱敏简述)5,200 kg/yr
25 kg 桶
25 kg
US$ 210-320 / kg
Qualified Partner — East China API Works
Entecavir INT-1|嘌呤核苷中间体
CAS 142217-80-9 · Antivirals
Target drug: entecavir
≥99.0%
单杂 ≤0.10%(脱敏)
糖苷化 + 保护基策略(脱敏简述)1,800 kg/yr
CEPUS DMFEU GMP
5 kg / 25 kg 桶
5 kg
US$ 1,150-1,700 / kg
Qualified Partner — East China API Works
Belzutifan INT-1|(R)-3-氟-5-[(茚满酮基)氧基]苯甲腈
CAS 2738675-96-0 · Anti-cancer
Target drug: belzutifan
高保密
≥99.0%
手性纯度 ≥99.5% ee(脱敏)
手性还原 + 成醚(脱敏简述)800 kg/yr
US DMF
1 kg / 5 kg 铝瓶
1 kg
US$ 3,400-4,900 / kg
Unibest Taizhou GMP-like Site
Belzutifan INT-2|3-[(茚满酮基)氧基]-5-氟苯甲腈
CAS 1672665-55-2 · Anti-cancer
Target drug: belzutifan
高保密
≥99.0%
单杂 ≤0.10%(脱敏)
成醚 + 砜基氧化(脱敏简述)1,100 kg/yr
5 kg 桶
2 kg
US$ 2,100-3,100 / kg
Unibest Taizhou GMP-like Site
2'-dG(iBu) 亚磷酰胺单体
CAS 68892-42-2 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)400 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,600-2,400 / 100g
Unibest Nantong cGMP Site
2'-dA(Bz) 亚磷酰胺单体
CAS 4546-72-9 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)400 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,480-2,200 / 100g
Unibest Nantong cGMP Site
2'-dC(Bz) 亚磷酰胺单体
CAS 4836-13-9 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)350 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,520-2,280 / 100g
Unibest Nantong cGMP Site

Official Intermediate Full CatalogWith CAS numbers · Aggregated by target drug

Total 493 intermediates · covering 255 target drugs
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