Unibest 优贝德

Cardiovascular / Renal Intermediates Catalogue58 intermediate products · 9 target APIs

Hypertension, heart failure, anticoagulation, chronic kidney disease

Classes follow the target API's primary indication (explicit mapping + catalogue links); unmapped targets are honestly shown as unclassified, never guessed.

Intermediate nameCAS No.Target drugAction
3-Chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one536760-29-9Apixaban
3-Morpholino-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one503615-03-0Apixaban
1-(4-Aminophenyl)-3-morpholino-5,6-dihydropyridin-2(1H)-one1267610-26-3Apixaban
3-Morpholino-1-[4-(2-oxopiperidin-1-yl)phenyl]-5,6-dihydropyridin.2(1H)-one545445-44-1Apixaban
Ethyl chloro[(4-methoxyphenyl)hydrazono]acetate27143-07-3Apixaban
1-(4-Methoxyphenyl)-7-0xo-6-[4-(2-0xopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acidethyl ester503614-91-3Apixaban
4-Bromo-2-methoxybenzaldehyde43192-33-2Finerenone
4-formyl-3-methoxybenzonitrile21962-45-8Finerenone
4-AMino-5-Methylpyridin-2-ol95306-64-2Finerenone
2-chloro-5-methylpyridin-4-amine79055-62-2Finerenone
2-Cyanoethyl 3-oxobutanoate65193-87-5Finerenone
2-cyanoethyl 4-(4-cyano-2-methoxyphenyl)-2,8-dimethyl-5-oxo-1,4,5,6-tetrahydro-1,6-naphthyridine-3-carboxylate1050477-43-4Finerenone
(R)-2-methylbut-3-enoic acid20626-49-7Milvexian
(5R,9S)-9-amino-21-(difluoromethyl)-5-methyl-21H-3-aza-1(4,2)-pyridina-2(5,4)-pyrazolacyclononaphan-4-one1802431-24-8Milvexian
6-(5-chloro-2-(4-chloro-1H-1,2,3-triazol-1-yl)phenyl)pyrimidin-4-ol1802430-55-2Milvexian
Pyrimidine, 4-[5-chloro-2-[4-(trimethylsilyl)-1H-1,2,3-triazol-1-yl]phenyl]-6-methoxy-1802430-53-0Milvexian
Pyrimidine, 4-[5-chloro-2-(4-chloro-1H-1,2,3-triazol-1-yl)phenyl]-6-methoxy-1802430-54-1Milvexian
tert-butyl(S)-(1-(4-chloropyridin-2-yl)but-3-en-1-yl)carbamate1329171-69-8Milvexian
Paricalcitol131918-61-1Paricalcitol
(1R,3aR,7aR)-1-((2R,5S,E)-6-hydroxy-5,6-diMethylhept-3-en-2-yl)-7a-Methylhexahydro-1H-inden-4(2H)-one95716-68-0Paricalcitol
(3R-trans)-[2-[3,5-Bis[[(1,1-diMethylethyl)diMethylsilyl]oxy]cyclohexylidene]ethyl]diphenyl-phosphine Oxide139356-39-1Paricalcitol
(1R,3aR,7aR)-1-((2R,5S,E)-6-(MethoxyMethoxy)-5,6-diMethylhept-3-en-2-yl)-7a-Methylhexahydro-1H-inden-4(2H)-one100858-26-2Paricalcitol
(((1R,3R)-5-((E)-2-((1R,3aS,7aR)-1-((2R,5S,E)-6-(MethoxyMethoxy)-5,6-diMethylhept-3-en-2-yl)-7a-Methylhexahydro-1H-inden-4(2H)-ylidene)ethylidene)cyclohexane-1,3-diyl)bis(oxy))bis(tert-butyldiMethylsilane)1435939-17-5Paricalcitol
(1R,3R)-5-((E)-2-((1R,3aS,7aR)-1-((2R,5S,E)-6-(MethoxyMethoxy)-5,6-diMethylhept-3-en-2-yl)-7a-Methyldihydro-1H-inden-4(2H,5H,6H,7H,7aH)-ylidene)ethylidene)cyclohexane-1,3-diol1023889-38-4Paricalcitol
tert-butyl 2-(4-amino-6-chloropyrimidin-5-yloxy)ethylmethylcarbamate1787294-51-2Treprostinil
4-(4-Aminophenyl)morpholin -3-one438056-69-0Rivaroxaban
(S)-(+)-N-(2,3-Epoxypropyl)phthalimide161596-47-0Rivaroxaban
5-Chlorothiophene-2-carboxylic acid24065-33-6Rivaroxaban
5-Chlorothiophene-2-carbonyl chloride42518-98-9Rivaroxaban
2-[[(5S)-2-0x0-3-[4-(3-0xo-4-morpholinyl)phenyl]-5-oxazolidinyl]methyl]-1H-isoindole-1,3(2H)-dione446292-08-6Rivaroxaban
4-[4-[(5S)-5-(Aminomethyl)-2-0xo-3-oxazolidinyl]phenyl] -3-morpholinone hydrochloride898543-06-1Rivaroxaban
2-[(2R)-2-Hydroxy-3-[[4-(3-oxo-4-Morpho linyl)phenyl]aMino]propyl]-1H-isoindole-1 ,3(2H)-dione446292-07-5Rivaroxaban
4-hydroxy-1-methyl-7-phenoxy-3-Isoquinolinecarboxylic acid1421312-35-7Roxadustat
4-hydroxy-1-methyl-7-phenoxy-3-Isoquinolinecarboxylic acid1421312-35-7Roxadustat
Methyl 4-hydroxy-7-phenoxyisoquinoline-3-carboxylate1455091-10-7Roxadustat
5-Phenoxyisobenzofuran-1(3H)-one57830-14-5Roxadustat
4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid ethyl ester1809286-36-9Roxadustat
4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid methyl ester1421312-34-6Roxadustat
(2-(N-(4,5-dimethylisoxazol-3-yl)-N-(methoxymethyl)sulfamoyl)phenyl)boronic acid415697-58-4Sparsentan
N-(4,5-dimethylisoxazol-3-yl)-N-(methoxymethyl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzenesulfonamide415697-56-2Sparsentan
4-bromo-3-(ethoxymethyl)benzaldehyde837408-71-6Sparsentan
4-bromo-3-ethoxymethyl-benzoic acid ethyl ester948349-66-4Sparsentan
N-(4,5-Dimethyl-3-isoxazolyl)-2'-(ethoxymethyl)-4'-formyl-N-(methoxymethyl)[1,1'-biphenyl]-2-sulfonamide1026913-68-7Sparsentan
N-(4,5-dimethylisoxazol-3-yl)-2'-(ethoxymethyl)-4'-(hydroxymethyl)-N-(methoxymethyl)-[1,1'-biphenyl]-2-sulfonamide1098924-76-5Sparsentan
4,6-Dichloro-2-(propylthio)pyrimidin -5-amine145783-15-9Ticagrelor
2-((3aR,4S,6R,6aS)-6-amino-2,2-dimethyltetrahydro -3aH-cyclopenta[d][1,3]dioxol -4-yloxy)ethanol L-tataric acid376608-65-0Ticagrelor
(1R,2S)-2-(3,4-Difluorophenyl)cyclopropanaminium(2R)hydroxy(phenyl)ethanoate376608-71-8Ticagrelor
Ethanol, 2-[[(3aR,4S,6R,6aS)-6-[[5-aMino-6-chloro-2-(propylthio)-4-pyriMidinyl]aMino]tetrahydro-2,2-diMethyl-4H-cyclopenta-1,3-dioxol-4-yl]oxy]-376608-74-1Ticagrelor
(1R,2S)-2-(3,4-difluorophenyl)cyclopropanamine hydrochloride1156491-10-9Ticagrelor
Cyclopropanamine,2-(3,4-difluorophenyl)-(1R,2S) -(2R,3R)-2,3-dihydroxybutanedioate (1:1)220352-39-6Ticagrelor
2-[[(3aS,4R,6S,6aR)-4-[7-[[(1R,2S)-2-(3,4-Difluorophenyl)cyclopropyl]amino]-5-(propylthio)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]-2,2-dimethyl-tetrahydro-3aH-cyclopenta[d][1,3]dioxol-6-yl]oxy]ethanol274693-26-4Ticagrelor
(1R,2R,3aS,9aS)-2,3,3a,4,9,9a-Hexahydro-1-[(3S)-3-hydroxyoctyl]-1H-benz[f]indene-2,5-diol101692-02-8Treprostinil
1-broMo-5-fluoro-2-Methyl-3-nitrobenzene502496-33-5Treprostinil
methyl 4-cyclopropyl-2-fluorobenzoate1613413-65-2Treprostinil
tert-butyl 2-(4-amino-6-chloropyrimidin-5-yloxy)ethylmethylcarbamate1787294-51-2Treprostinil
2H-Benz[f]inden-2-one, 9-[[(1,1-dimethylethyl)dimethylsilyl]oxy]-3,3a,4,9-tetrahydro-5-methoxy-1-[(3S)-3-[(tetrahydro-2H-pyran-2-yl)oxy]octyl]-, (3aS,9R)-223734-60-9Treprostinil
2-allyl-3-methoxybenzaldehyde94956-98-6Treprostinil
(5S)-1-Decyn-5-ol848609-05-2Treprostinil

The catalogue keeps growing; use RFQ for quotes or complex programmes.