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Lascufloxacin

Tier C — Watch / trade

Lascufloxacin

Kyorin Pharmaceutical Co Ltd
Originator
2019
First approval
-
Expiry (public)
$0.02B ▲
Peak sales
化学药
Type

TargetsTopoisomerase IV、Bacterial DNA gyrase

BrandLasvic

Indications (approved)耳鼻咽喉疾病、肺炎、呼吸道感染

Regional status

US
-
EU
-
China
-
Japan
批准上市
2019-09-20

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 5 · Total yield 9.57 kg
Synthetic routes & intermediates Route 1
CodeCAS No.Intermediate
LASC-001635319-09-4tert-butyl (3R,4R)-3-hydroxy-4-(hydroxymethyl)pyrrolidine-1-carboxylate
LASC-002848416-47-7tert-butyl (3S,4R)-3-(bromomethyl)-4-hydroxypyrrolidine-1-carboxylate
LASC-003848416-48-8tert-butyl (3S,4S)-3-(bromomethyl)-4-fluoropyrrolidine-1-carboxylate
LASC-004848416-49-9tert-butyl (3S,4S)-3-((cyclopropylamino)methyl)-4-fluoropyrrolidine-1-carboxylate
LASC-005604798-54-1N-(((3R,4S)-4-fluoropyrrolidin-3-yl)methyl)cyclopropanamine
LASC-006848498-67-98,9-difluoro-6-(2-fluoroethyl)-7-methoxy-4-oxo-4,6-dihydro-2H-1l3,2l4-[1,3,2]dioxaborinino[5,6-c]quinoline-2,2-diyl diacetate

Frequently asked questions

What are the approved indications of Lascufloxacin?

Approved indications include: 耳鼻咽喉疾病, 肺炎, 呼吸道感染.

When does the Lascufloxacin patent expire?

No public expiry year is available for Lascufloxacin yet; this page updates once verified.

How many synthesis routes are recorded for Lascufloxacin?

1 synthesis routes are recorded; the shortest is 5 steps with 9.57 kg total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Lascufloxacin intermediates?

All intermediates in Lascufloxacin routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Lascufloxacin intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-24