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Conteltinib

Tier C — Watch / trade

Conteltinib

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Originator
2026
First approval
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Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:IGF1R, ALK, FAK1, FAK2

Indications (approved):Non-small cell lung cancer

Regional status

US
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EU
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China
Approved
2026-06-10
Japan
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Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 11 · Total yield 685 g
Conteltinib-001873-83-6Conteltinib-002107-20-0Conteltinib-00339929-79-8Conteltinib-00416372-12-6Conteltinib-0052139336-89-1Conteltinib-0061312162-73-4Conteltinib-00779099-07-3Conteltinib-008109-01-3Conteltinib-009190964-91-1Conteltinib-01053617-36-0Conteltinib-011448-19-1Conteltinib-012761440-65-7Conteltinib-013761440-75-9Conteltinib-014109-86-4Conteltinib-0152139336-90-4Conteltinib-016761435-31-8Conteltinib-0172139336-91-5API · Conteltinib
CodeCAS No.Intermediate
Conteltinib-001873-83-66-aminopyrimidine-2,4(1H,3H)-dione
Conteltinib-002107-20-02-chloroacetaldehyde
Conteltinib-00339929-79-87H-pyrrolo[2,3-d]pyrimidine-2,4-diol
Conteltinib-00416372-12-66,7-dihydro-5H-pyrrolo[2,3-d]pyrimidine-2,4-diol
Conteltinib-0052139336-89-12,4-dichloro-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidine
Conteltinib-0061312162-73-42,4-dichloro-7-(4-methoxybenzyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidine
Conteltinib-00779099-07-3tert-butyl 4-oxopiperidine-1-carboxylate
Conteltinib-008109-01-3Available1-methylpiperazine
Conteltinib-009190964-91-1tert-butyl 4-(4-methylpiperazin-1-yl)piperidine-1-carboxylate
Conteltinib-01053617-36-01-methyl-4-(piperidin-4-yl)piperazine
Conteltinib-011448-19-14-fluoro-2-methoxy-1-nitrobenzene
Conteltinib-012761440-65-71-(1-(3-methoxy-4-nitrophenyl)piperidin-4-yl)-4-methylpiperazine
Conteltinib-013761440-75-9Available2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)aniline
Conteltinib-014109-86-42-methoxyethan-1-ol
Conteltinib-0152139336-90-44-chloro-N-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)-7-(4-methoxybenzyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-2-amine
Conteltinib-016761435-31-82-amino-N-isopropylbenzenesulfonamide
Conteltinib-0172139336-91-5N-isopropyl-2-((2-((2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)amino)-7-(4-methoxybenzyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)benzenesulfonamide

Frequently asked questions

What are the approved indications of Conteltinib?

Approved indications include: Non-small cell lung cancer.

When does the Conteltinib patent expire?

No public expiry year is available for Conteltinib yet; this page updates once verified.

How many synthesis routes are recorded for Conteltinib?

1 synthesis routes are recorded; the shortest is 11 steps with 685 g total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Conteltinib intermediates?

2 intermediate CAS of Conteltinib are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Conteltinib intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-27