Umirolimus
Tier C — Watch / tradeUmirolimus
Targets：mTOR
Brand：LUMENO、Nobori
Indications (approved)：冠状动脉再狭窄
Regional status
Synthetic routes & intermediates2 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| Umirolimus-001 | 110-80-5 | 2-Ethoxyethanol |
| Umirolimus-002 | 832-53-1 | 2,3,4,5,6-Pentafluorobenzenesulfonyl chloride |
| Umirolimus-003 | 1196708-70-9 | Pentafluorobenzenesulfonic acid 2-ethoxyethyl ester |
| Umirolimus-004 | 53123-88-9 | (3S,6R,7E,9R,10R,12R,14S,15E,17E,19E,21S,23S,26R,27R,34aS)-9,27-Dihydroxy-3-[1-[(1S,3R,4R)-4-hydroxy-3-methoxycyclohexyl]propan-2(R)-yl]-10,21-dimethoxy-6,8,12,14,20,26-hexamethyl-3,4,5,6,9,10,11,12,13,14,21,22,23,24,25,26,27,28,29,31,32,33,34,34a-tetracosahydro-1H-23,27-epoxypyrido[2,1-c][1,4]oxazacyclohentriacontine-1,5,11,28,29(4H,6H,31H)-pentone |
| Code | CAS No. | Intermediate |
|---|---|---|
| Umirolimus-001 | 110-80-5 | 2-Ethoxyethanol |
| Umirolimus-005 | 17178-12-0 | 2-Ethoxyethyl 4-chlorobenzenesulfonate |
| Umirolimus-006 | 851536-76-0 | 2-Ethoxyethyl trifluoromethanesulfonate |
| Umirolimus-004 | 53123-88-9 | (3S,6R,7E,9R,10R,12R,14S,15E,17E,19E,21S,23S,26R,27R,34aS)-9,27-Dihydroxy-3-[1-[(1S,3R,4R)-4-hydroxy-3-methoxycyclohexyl]propan-2(R)-yl]-10,21-dimethoxy-6,8,12,14,20,26-hexamethyl-3,4,5,6,9,10,11,12,13,14,21,22,23,24,25,26,27,28,29,31,32,33,34,34a-tetracosahydro-1H-23,27-epoxypyrido[2,1-c][1,4]oxazacyclohentriacontine-1,5,11,28,29(4H,6H,31H)-pentone |
Frequently asked questions
What are the approved indications of Umirolimus?
Approved indications include: 冠状动脉再狭窄.
When does the Umirolimus patent expire?
No public expiry year is available for Umirolimus yet; this page updates once verified.
How many synthesis routes are recorded for Umirolimus?
2 synthesis routes are recorded; the shortest is 2 steps with 0.498g(Umirolimus (Free)) total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Umirolimus intermediates?
All intermediates in Umirolimus routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.
How do I get a quote for Umirolimus intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-09-24