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Glycopyrrolate Tosylate

Tier C — Watch / trade

Glycopyrrolate Tosylate

Dermira Inc
Originator
2018
First approval
-
Expiry (public)
No sales data
Peak sales
化学药
Type

TargetsmAChRs

BrandRapifort、Qbrexza

Indications (approved)多汗症

Regional status

US
批准上市
2018-06-28
EU
无进展
2015-03-30
China
无进展
2015-03-30
Japan
批准上市
2022-01-20

Synthetic routes & intermediates2 routes

Originator routes × 0Optimised (non-patent) × 2Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 4 · Total yield /
Synthetic routes & intermediates Route 1
CodeCAS No.Intermediate
(I)860865-1-a427-49-6(+/-)-Cyclopentylmandelic acid
(II)860865-1-a1246930-41-52-Cyclopentyl-2-hydroxy-1-(1H-imidazol-1-yl)-2-phenylethanone
(III)860865-1-a13220-33-21-Methylpyrrolidin-3-ol
(IV)860865-1-a13118-11-1(1-Methylpyrrolidin-3-yl) 2-cyclopentyl-2-hydroxy-2-phenylacetate
(V)860865-1-a-(3R)-1-Methylpyrrolidin-3-yl (2S)-cyclopentyl(hydroxy)phenylacetate
(VI)860865-1-a80-48-84-Methylbenzenesulfonic acid methyl ester
OptimisedRoute 2Steps 1 · Total yield /
Synthetic routes & intermediates Route 2
CodeCAS No.Intermediate
(Ia)860865-2-a-3(R*)-[2(S*)-Cyclopentyl-2-hydroxy-2-phenylacetyloxy]-1,1-dimethylpyrrolidinium bromide
(Ib)860865-2-a-(3R)-3-[[(2S)-2-Cyclopentyl-2-hydroxy-2-phenylacetyl]oxy]-1,1-dimethylpyrrolidin-1-ium acetate

Frequently asked questions

What are the approved indications of Glycopyrrolate Tosylate?

Approved indications include: 多汗症.

When does the Glycopyrrolate Tosylate patent expire?

No public expiry year is available for Glycopyrrolate Tosylate yet; this page updates once verified.

How many synthesis routes are recorded for Glycopyrrolate Tosylate?

2 synthesis routes are recorded; the shortest is 1 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Glycopyrrolate Tosylate intermediates?

All intermediates in Glycopyrrolate Tosylate routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Glycopyrrolate Tosylate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-24