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CAS 59858-41-2

2-(Diethylamino)acetyl chloride

Codes:Lidocaine Hydrochloride-012

Application context (from source-drug indications)

早泄利多卡因/丙胺卡因皮肤气雾剂生理性性功能障碍利多卡因/丙胺卡因皮肤气雾剂滴虫感染咪康唑/甲硝唑/利多卡因念珠菌病咪康唑/甲硝唑/利多卡因阴道炎咪康唑/甲硝唑/利多卡因

Source drugs (routes using this intermediate)

DrugTierExpiry
利多卡因/丙胺卡因皮肤气雾剂Lidocaine/Prilocaine cutaneous sprayTier C — Watch / trade-
咪康唑/甲硝唑/利多卡因Miconazole/Metronidazole/LidocaineTier C — Watch / trade-

Position in synthesis routes (up/downstream chain)

Ordered by route registration; left → right is the synthesis direction. The highlighted node is the current CAS; others link to their own profiles.

利多卡因/丙胺卡因皮肤气雾剂工艺路线steps: 8total yield: 93.4kg(Lidocaine Hydrochloride (API))
1,3-Dimethyl-2-nitrobenzene→2-Amino-1,3-dimethylbenzene→2-Bromanylethanoic acid→2-Chloroacetic acid→2-Chloranylethanoyl chloride→2-Chloroacetic acid methyl ester→2-Bromo-N-(2,6-dimethylphenyl)acetamide→1-Chloroacetylamino-2,6-dimethylbenzene→N-Ethylethanamine→2-Diethylamino-N-(2,6-dimethylphenyl)acetamide→2-(Diethylamino)acetic acid→2-(Diethylamino)acetyl chloride→Methyl 2-(diethylamino)acetate→3-(2-Methoxyphenyl)-1H-pyrazole→2-(Chloromethyl)pyridine hydrochloride→Lidocaine Hydrochloride-016→Dichloridomanganese 2-[[3-(2-methoxyphenyl)-1H-pyrazol-1-yl]methyl]pyridine
咪康唑/甲硝唑/利多卡因工艺路线steps: 8total yield: 93.4kg(Lidocaine Hydrochloride (API))
1,3-Dimethyl-2-nitrobenzene→2-Amino-1,3-dimethylbenzene→2-Bromanylethanoic acid→2-Chloroacetic acid→2-Chloranylethanoyl chloride→2-Chloroacetic acid methyl ester→2-Bromo-N-(2,6-dimethylphenyl)acetamide→1-Chloroacetylamino-2,6-dimethylbenzene→N-Ethylethanamine→2-Diethylamino-N-(2,6-dimethylphenyl)acetamide→2-(Diethylamino)acetic acid→2-(Diethylamino)acetyl chloride→Methyl 2-(diethylamino)acetate→3-(2-Methoxyphenyl)-1H-pyrazole→2-(Chloromethyl)pyridine hydrochloride→Lidocaine Hydrochloride-016→Dichloridomanganese 2-[[3-(2-methoxyphenyl)-1H-pyrazol-1-yl]methyl]pyridine

Intermediates available on this site

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This is a CAS-level registry record: registrations across routes are merged. Supplier offers and buyer demands will be matched on this CAS as the primary key.