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CAS 112914-13-3
[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine
登记编号：Mosapride Citrate-006
应用背景（按来源药适应症）
胃炎枸橼酸莫沙必利肠内喂养不耐受枸橼酸莫沙必利肠易激综合征枸橼酸莫沙必利消化不良枸橼酸莫沙必利便秘枸橼酸莫沙必利
来源药（使用该中间体的合成路线）
| 品种 | 梯队 | 到期年 |
|---|---|---|
| 枸橼酸莫沙必利Mosapride Citrate | Tier C · 观察 / 贸易 | - |
合成路线中的位置（上下游链）
按路线登记顺序排列，左→右为合成方向；高亮为当前 CAS，其余可点击跳转对应档案。
Methyl 4-(acetylamino)-2-hydroxybenzoate→1-Iodoethane→methyl 4-acetamido-2-ethoxybenzoate→methyl 5-chloro-4-acetamido-2-ethoxybenzoate→4-Amino-5-chloro-2-ethoxybenzoic acid→[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine→Mosapride Citrate-007
[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine→Sulfuric acid 1-[4-[(4-fluorophenyl)methyl]morpholin-2-yl]methanamine→Phosphoric acid 1-[4-[(4-fluorophenyl)methyl]morpholin-2-yl]methanamine→1-[4-[(4-Fluorophenyl)methyl]morpholin-2-yl]methanamine hydrogen chloride→2-Methylpropane-1,2,3-tricarboxylic acid 1-[4-[(4-fluorophenyl)methyl]morpholin-2-yl]methanamine→4-Fluorobenzaldehyde→2-Hydroxyethylamine→2-[(E)-[(4-Fluorophenyl)methylidene]amino]ethan-1-ol→2-[[(4-Fluorophenyl)methyl]amino]ethan-1-ol→2-[(Oxiran-2-yl)methyl]-1H-isoindole-1,3(2H)-dione→1,3-Dihydro-1,3-dioxoisoindole→1,3-Dihydro-1,3-dioxoisoindole potassium salt→(+/-)-Epichlorohydrin
[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine→2-Hydroxyethylamine→2-[[(4-Fluorophenyl)methyl]amino]ethan-1-ol→1,3-Dihydro-1,3-dioxoisoindole potassium salt→Glycerol-alpha,gamma-dichlorohydrin→N-(3-Chloro-2-hydroxypropyl)-phthalimide→2-(3-[[(4-Fluorophenyl)methyl](2-hydroxyethyl)amino]-2-hydroxypropyl)-1H-isoindole-1,3(2H)-dione→2-[2-Hydroxy-3-[(2-hydroxyethyl)amino]propyl]-1H-isoindole-1,3(2H)-dione→Morpholin-2-ylmethanamine→alpha-Chloro-4-fluorotoluene
4-amino-5-chloro-2-ethoxy-3-hydroxy-N-[(5-oxomorpholin-2-yl)methyl]benzamide→4-amino-5-chloro-2-ethoxy-3-hydroxy-N-(morpholin-2-ylmethyl)benzamide→2,3-Dihydroxybenzaldehyde→2-ethoxy-3-hydroxybenzaldehyde→2-ethoxy-3-hydroxy-4-nitrobenzaldehyde→2-ethoxy-3-hydroxy-4-nitrobenzoic acid→6-(aminomethyl)morpholin-3-one→2-ethoxy-3-hydroxy-4-nitro-N-[(5-oxomorpholin-2-yl)methyl]benzamide→4-amino-2-ethoxy-3-hydroxy-N-[(5-oxomorpholin-2-yl)methyl]benzamide→2-ethoxy-3-hydroxy-4-nitrobenzoyl chloride→[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine→2-ethoxy-N-({4-[(4-fluorophenyl)methyl]morpholin-2-yl}methyl)-3-hydroxy-4-nitrobenzamide→tert-butyl 2-{[(2-ethoxy-3-hydroxy-4-nitrophenyl)formamido]methyl}morpholine-4-carboxylate→tert-butyl 2-{[(4-acetamido-2-ethoxy-3-hydroxyphenyl)formamido]methyl}morpholine-4-carboxylate→tert-butyl 2-{[(5-chloro-4-acetamido-2-ethoxy-3-hydroxyphenyl)formamido]methyl}morpholine-4-carboxylate
2-Fluoro-4-nitrobenzenecarboxylic acid→Methyl 2-fluoro-4-nitrobenzenecarboxylate→Ethanol sodium salt→Methyl 2-ethoxy-4-nitrobenzoate→Methyl 5-chloro-2-ethoxy-4-nitrobenzoate→[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine→Mosapride Citrate-007
1-Chloro-2-methylbenzene→2-Chloro-1-methyl-4-nitrobenzene→Potassium ethanolate→2-Ethoxy-1-methyl-4-nitrobenzene→1-(Bromomethyl)-2-ethoxy-4-nitrobenzene→1-(Bromomethyl)-5-chloro-2-ethoxy-4-nitrobenzene→1-Chloro-4-ethoxy-5-(methoxymethyl)-2-nitrobenzene→2-Chloro-5-ethoxy-4-(methoxymethyl)aniline→[4-(4-Fluorobenzyl)-2-morpholinyl]methylamine→Mosapride Citrate-007
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