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Pharmaceutical Intermediates

Full official intermediate catalog + key intermediates with CEP / DMF / GMP / cold-chain qualifications and capacity details · each quotable via RFQ

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Orforglipron intermediates

样品订单(各 500g)+ 0.5KG 复购

2 deals completed · latest 2026-09-21

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PINACOLONE

两用物项贸易品类

2 deals completed · latest 2026-01-19

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4-(3-Bromophenyl)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline

CAS 543737-10-6

1 deal completed · latest 2026-07-08

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By Therapeutic Area of Target Drug

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Official Intermediate Full CatalogWith CAS numbers · Aggregated by target drug

Total 193 intermediates · covering 255 target drugs
Intermediate nameCAS No.Target drugAction
(S)-3-(5-bromo-1-ethyl-2-(2-(1-methoxyethyl)pyridin-3-yl)-1H-indol-3-yl)-2,2-dimethylpropan-1-ol2641820-94-0RMC6236 Daraxonrasib
(S)-3-bromo-2-(1-methoxyethyl)pyridine641451-44-5RMC6236 Daraxonrasib
(S)-3-bromo-2-(1-methoxyethyl)pyridine641451-44-5RMC6236 Daraxonrasib
3,3-dimethyldihydro-2H-pyran-2,6(3H)-dione2938-48-9RMC6236 Daraxonrasib
3,3-dimethyldihydro-2H-pyran-2,6(3H)-dione2938-48-9RMC6236 Daraxonrasib
ethyl (S)-3-(5-bromo-2-(2-(1-methoxyethyl)pyridin-3-yl)-1H-indol-3-yl)-2,2-dimethylpropanoate2641451-50-3RMC6236 Daraxonrasib
methyl (R)-2-((tert-butoxycarbonyl)amino)-3-iodopropanoate93267-04-0RMC6236 Daraxonrasib
methyl (R)-2-((tert-butoxycarbonyl)amino)-3-iodopropanoate93267-04-0RMC6236 Daraxonrasib
Methyl (S)-1-((S)-3-(4-bromothiazol-2-yl)-2-((1S,2S)-2-methylcyclopropane-1-carboxamido)propanoyl)Hexahydropyridazine-3-carboxylate3060084-27-4RMC6236 Daraxonrasib
Methyl (S)-hexahydropyridazine-3-carboxylate hydrochloride380223-17-6RMC6236 Daraxonrasib
-CYCLOPENTYLACRYLONITRILE591769-05-0Ruxolitinib phosphate
(3R)-3-cyclopentyl-3-[4-(7-[2-(trimethylsilyl)ethoxy]methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile941685-40-1Ruxolitinib phosphate
(4-(1-(2-Cyano-1-cyclopentylethyl)-1h-pyrazol-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl)methyl pivalate1236033-05-8Ruxolitinib phosphate
(4-Chloro-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl pivalate1146629-75-5Ruxolitinib phosphate
(R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile41678-49-5Ruxolitinib phosphate
(R)-3-(4-broMo-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile1146629-83-5Ruxolitinib phosphate
(R)-3-cyclopentyl-3-(4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)propanenitrile1146629-84-6Ruxolitinib phosphate
(S)-3-cyclopentyl-3-hydrazinylpropanenitrile L-tartaric acid salt dihydrate2761879-36-9Ruxolitinib phosphate
1-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole1029716-44-6Ruxolitinib phosphate
1-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole1029716-44-6Ruxolitinib phosphate
1H-Pyrazole-1-propanamide, 4-bromo-β-cyclopentyl-, (βR)-2201066-06-8Ruxolitinib phosphate
2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)acetic acid1000518-93-3Ruxolitinib phosphate
3-Cyclopentyl-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]propanenitrile1153949-38-2Ruxolitinib phosphate
3-cyclopentyl-3-[4-(7-[2-(trimethylsilyl)ethoxy]methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile941685-39-8Ruxolitinib phosphate
4-(1H-pyrazol-4-yl)-7-((2-(trimethylsilyl)ethoxy)methyl)-7H-pyrrolo[2,3-d]pyrimidine941685-27-4Ruxolitinib phosphate
4-CHLORO-7-((2-(TRIMETHYLSILYL)ETHOXY)METHYL)-7H-PYRROLO[2,3-D]PYRIMIDINE941685-26-3Ruxolitinib phosphate
4-Chloropyrrolo[2,3-d]pyrimidine3680-69-1Ruxolitinib phosphate
4-methyl-7H-pyrrolo[2,3-d]pyrimidine945950-37-8Ruxolitinib phosphate
Cyclopentanecarbaldehyde872-53-7Ruxolitinib phosphate
1-Aminopyrazin-1-ium 2,4,6-trimethylbenzenesulfonat57489-85-7 Saracatinib
2-Fluoropyridine-5-boronic acid pinacol ester444120-95-0Saracatinib
6-Bromo-4-hydroxy-pyrazolo[1,5-a]pyridine-3-carbonitrile2068065-16-5Saracatinib
6-bromo-4-methoxypyrazolo[1,5-a]pyridine-3-carbonitrile1207836-10-9Saracatinib
6-Methoxynicotinaldehyde65873-72-5Saracatinib
N-Phenyl-bis(trifluoromethanesulfonimide)37595-74-7Saracatinib
Tert-butyl 3,6-diazabicyclo[3.1.1]heptane-6-carboxylate869494-16-6Saracatinib
(S)-4-N-Boc-2-methylpiperazine147081-29-6Sotorasib
2-Fluoro-6-hydroxybenzeneboronic acid pinacol ester1534369-41-9Sotorasib
2-Fluoro-6-methoxyphenylboronic acid78495-63-3Sotorasib
2,6-Dichloro-5-fluoronicotinamide113237-20-0Sotorasib
4-[(S)-4-Boc-2-methyl-1-piperazinyl]-6-fluoro-7-(2-fluoro-6-hydroxyphenyl)-1-(2-isopropyl-4-methyl-3-pyridyl)pyrido[2,3-d]pyrimidin-2(1H)-one2252403-85-1Sotorasib
7-chloro-6-fluoro-1-(2-isopropyl-4-methylpyridin-3-yl)pyrido[2,3-d]pyrimidine-2,4(1H,3H)-dione2300966-23-6Sotorasib
7-chloro-6-fluoro-1-(2-isopropyl-4-methylpyridin-3-yl)pyrido[2,3-d]pyrimidine-2,4(1H,3H)-dione2300966-23-6Sotorasib
Fluoro-6-hydroxyphenylboronic acid1256345-60-4Sotorasib
isopropyl-4-methylpyridin-3-amine1698293-93-4Sotorasib
Potassium Trifluoro(2-fluoro-6-hydroxyphenyl)borate2252415-10-2Sotorasib
tert-butyl (S)-4-(7-chloro-6-fluoro-1-(2-isopropyl-4-methylpyridin-3-yl)-2-oxo-1,2-dihydropyrido[2,3-d]pyrimidin-4-yl)-3-methylpiperazine-1-carboxylate2252403-84-0Sotorasib
[1,1'-Biphenyl]-3-carboxylic acid, 5-[ethyl(tetrahydro-2H-pyran-4-yl)amino]-4-methyl-4'-(4-morpholinylmethyl)-1403259-00-6Tazemetostat Hydrobromide
[1,1'-Biphenyl]-3-carboxylic acid, 5-[ethyl(tetrahydro-2H-pyran-4-yl)amino]-4-methyl-4'-(4-morpholinylmethyl)-, methyl ester1403258-99-0Tazemetostat Hydrobromide
3-(aminomethyl)-4,6-dimethyl-1,2-dihydropyridin-2-one hydrochloride1173081-96-3Tazemetostat Hydrobromide
4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)morpholine364794-79-6Tazemetostat Hydrobromide
5-Bromo-2-methyl-3-nitrobenzoic acid107650-20-4Tazemetostat Hydrobromide
Methyl 3-amino-5-bromo-2-methylbenzoate1000342-11-9Tazemetostat Hydrobromide
Methyl 5-bromo-2-methyl-3-((tetrahydro-2H-pyran-4-yl)amino)benzoate1403257-49-7Tazemetostat Hydrobromide
Methyl 5-bromo-2-methyl-3-nitrobenzoate220514-28-3Tazemetostat Hydrobromide
Methyl 5-bromo-3-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-2-methylbenzoate1403257-79-3Tazemetostat Hydrobromide
(2-methyl-4-nitrophenoxy)-[1,2,4]triazolo[1,5-a]pyridine937263-44-0Tucatinib
(4-chloropyridin-2-yl)-N'-hydroxyformimidamide2379814-46-5Tucatinib
(E)-N'-(2-cyano-4-(3-(1-hydroxy-2-methylpropan-2-yl)thioureido)phenyl)-N,N-dimethylformimidamide1429755-57-6Tucatinib
(E)-N'-(2-cyano-4-nitrophenyl)-N,N-dimethylformimidamide39263-34-8Tucatinib