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氟贝他吡[18F]

Tier C — Watch / trade

Florbetapir(18F)

礼来制药
Originator
2012
First approval
-
Expiry (public)
No sales data
Peak sales
放射性产品
Type

TargetsAPP

BrandAmyvid、艾美维

Indications (approved)阿尔茨海默病、造影检查

Regional status

US
批准上市
2012-04-06
EU
批准上市
2013-01-14
China
批准上市
2025-06-03
Japan
批准上市
2016-12-19

Synthetic routes & intermediates1 routes

Originator routes × 0Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 6 · Total yield /
Synthetic routes & intermediates Route 1
CodeCAS No.Intermediate
FLORB-001112-27-62,2'-(ethane-1,2-diylbis(oxy))bis(ethan-1-ol)
FLORB-00273290-22-92-bromo-5-iodopyridine
FLORB-0031234208-03-72-(2-(2-((5-iodopyridin-2-yl)oxy)ethoxy)ethoxy)ethan-1-ol
FLORB-004937183-61-4tert-butyl methyl(4-vinylphenyl)carbamate
FLORB-0051234208-02-6tert-butyl (E)-(4-(2-(6-(2-(2-(2-hydroxyethoxy)ethoxy)ethoxy)pyridin-3-yl)vinyl)phenyl)(methyl)carbamate
FLORB-0061205550-99-7(E)-2-(2-(2-((5-(4-((tert-butoxycarbonyl)(methyl)amino)styryl)pyridin-2-yl)oxy)ethoxy)ethoxy)ethyl 4-methylbenzenesulfonate
FLORB-0071520-21-44-vinylaniline
FLORB-00857295-14-4tert-butyl (4-vinylphenyl)carbamate

Frequently asked questions

What are the approved indications of Florbetapir(18F)?

Approved indications include: 阿尔茨海默病, 造影检查.

When does the Florbetapir(18F) patent expire?

No public expiry year is available for Florbetapir(18F) yet; this page updates once verified.

How many synthesis routes are recorded for Florbetapir(18F)?

1 synthesis routes are recorded; the shortest is 6 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Florbetapir(18F) intermediates?

All intermediates in Florbetapir(18F) routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Florbetapir(18F) intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-24