门冬氨酸帕瑞肽
Tier C — Watch / tradePasireotide Diaspartate
Targets：SSTR3、SSTR1、SSTR5、SSTR2
Brand：丝尼芬、Signifor
Indications (approved)：库欣综合征、垂体ACTH分泌过多
Regional status
Synthetic routes & intermediates3 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| PASI-001 | - | - |
| PASI-002 | - | - |
| PASI-003 | - | - |
| PASI-004 | - | - |
| PASI-005 | - | - |
| PASI-006 | 187223-15-0 | (2S,4R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-(((2-((tert-butoxycarbonyl)amino)ethyl)carbamoyl)oxy)pyrrolidine-2-carboxylic acid |
| PASI-007 | - | - |
| PASI-008 | - | - |
| PASI-009 | - | - |
| PASI-010 | 1499-56-5 | (2S,4R)-methyl 4-hydroxypyrrolidine-2-carboxylate |
| PASI-011 | 122350-59-8 | 1-((9H-fluoren-9-yl)methyl) 2-methyl (2S,4R)-4-hydroxypyrrolidine-1,2-dicarboxylate |
| PASI-012 | 556796-28-2 | 1-((9H-fluoren-9-yl)methyl) 2-methyl (2S,4R)-4-((chlorocarbonyl)oxy)pyrrolidine-1,2-dicarboxylate |
| PASI-013 | 57260-73-8Available | tert-butyl (2-aminoethyl)carbamate |
| PASI-014 | 187223-14-9 | 1-((9H-fluoren-9-yl)methyl) 2-methyl (2S,4R)-4-(((2-((tert-butoxycarbonyl)amino)ethyl)carbamoyl)oxy)pyrrolidine-1,2-dicarboxylate |
| PASI-015 | 556796-29-3 | (2S,4R)-4-(((2-((tert-butoxycarbonyl)amino)ethyl)carbamoyl)oxy)pyrrolidine-2-carboxylic acid |
| Code | CAS No. | Intermediate |
|---|---|---|
| PASI-006 | 187223-15-0 | (2S,4R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-(((2-((tert-butoxycarbonyl)amino)ethyl)carbamoyl)oxy)pyrrolidine-2-carboxylic acid |
| PASI-016 | 187223-14-9 | 1-((9H-fluoren-9-yl)methyl) 2-methyl (2S,4R)-4-(((2-((tert-butoxycarbonyl)amino)ethyl)carbamoyl)oxy)pyrrolidine-1,2-dicarboxylate |
| PASI-017 | - | - |
| PASI-018 | - | - |
| PASI-019 | - | - |
| PASI-020 | - | - |
| PASI-021 | - | - |
| PASI-022 | 1527478-88-1 | - |
| PASI-023 | - | #N/A |
| Code | CAS No. | Intermediate |
|---|---|---|
| PASI-024 | - | (E)-prop-1-en-1-yl (((9H-fluoren-9-yl)methoxy)carbonyl)-L-lysinate |
| PASI-025 | - | - |
| PASI-026 | - | - |
| PASI-027 | - | - |
| PASI-028 | - | - |
| PASI-029 | 1427038-62-7 | (2-((tert-butoxycarbonyl)amino)ethyl)carbamic acid |
| PASI-030 | - | - |
| PASI-031 | - | - |
| PASI-032 | - | - |
| PASI-033 | - | - |
Frequently asked questions
What are the approved indications of Pasireotide Diaspartate?
Approved indications include: 库欣综合征, 垂体ACTH分泌过多.
When does the Pasireotide Diaspartate patent expire?
No public expiry year is available for Pasireotide Diaspartate yet; this page updates once verified.
How many synthesis routes are recorded for Pasireotide Diaspartate?
3 synthesis routes are recorded; the shortest is 9 steps with / total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Pasireotide Diaspartate intermediates?
1 intermediate CAS of Pasireotide Diaspartate are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.
How do I get a quote for Pasireotide Diaspartate intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-09-24