替戈拉生
Tier C — Watch / tradeTegoprazan
Targets：H+/K+ ATPase
Brand：K-Cab Tab、泰欣赞
Indications (approved)：胃食管反流病、幽门螺杆菌感染、十二指肠溃疡
Regional status
Synthetic routes & intermediates1 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| TEGO-001 | 713530-47-3Available | 2-(benzyloxy)-4-bromo-6-nitroaniline |
| TEGO-002 | 942195-80-4Available | N-(2-(benzyloxy)-4-bromo-6-nitrophenyl)acetamide |
| TEGO-003 | 942195-81-5Available | N-(2-(benzyloxy)-4-cyano-6-nitrophenyl)acetamide |
| TEGO-004 | 942195-82-6Available | 4-(benzyloxy)-2-methyl-1H-benzo[d]imidazole-6-carbonitrile |
| TEGO-005 | 942195-83-7Available | 4-(benzyloxy)-2-methyl-1H-benzo[d]imidazole-6-carboxylic acid |
| TEGO-006 | 942195-84-8Available | 4-(benzyloxy)-N,N,2-trimethyl-1H-benzo[d]imidazole-6-carboxamide |
| TEGO-007 | 942195-85-9Available | 4-(benzyloxy)-N,N,2-trimethyl-1-tosyl-1H-benzo[d]imidazole-6-carboxamide |
| TEGO-008 | 942195-86-0Available | 4-hydroxy-N,N,2-trimethyl-1-tosyl-1H-benzo[d]imidazole-6-carboxamide |
| TEGO-009 | 917248-51-2Available | 5,7-difluorochroman-4-ol |
| TEGO-010 | 942195-87-1Available | 4-((5,7-difluorochroman-4-yl)oxy)-N,N,2-trimethyl-1-tosyl-1H-benzo[d]imidazole-6-carboxamide |
| TEGO-011 | 942195-54-2Available | 4-((5,7-difluorochroman-4-yl)oxy)-N,N,2-trimethyl-1H-benzo[d]imidazole-6-carboxamide |
Frequently asked questions
What are the approved indications of Tegoprazan?
Approved indications include: 胃食管反流病, 幽门螺杆菌感染, 十二指肠溃疡.
When does the Tegoprazan patent expire?
No public expiry year is available for Tegoprazan yet; this page updates once verified.
How many synthesis routes are recorded for Tegoprazan?
1 synthesis routes are recorded; the shortest is 10 steps with 582 mg total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Tegoprazan intermediates?
11 intermediate CAS of Tegoprazan are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.
How do I get a quote for Tegoprazan intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-09-24