赛利司他

Tier C — Watch / trade

Cetilistat

Norgine Europe Bv

Originator

2013

First approval

Expiry (public)

No sales data

Peak sales

化学药

Type

Targets：LIPF

Brand：Oblean

Indications (approved)：肥胖症

Regional status

无进展

2005-04-01

无进展

2004-12-01

China

Japan

批准上市

2013-09-20

Synthetic routes & intermediates3 routes

Originator routes × 1Optimised (non-patent) × 2Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 2 · Total yield 2.51 g

Code	CAS No.	Intermediate
CETI-001	36653-82-4	hexadecan-1-ol
CETI-002	26272-90-2	hexadecyl carbonochloridate
CETI-003	2941-78-8	2-amino-5-methylbenzoic acid

OptimisedRoute 2Steps 4 · Total yield 3.3 g

Synthetic routes & intermediates Route 2

Code	CAS No.	Intermediate
CETI-001	36653-82-4	hexadecan-1-ol
CETI-004	622-58-2	1-isocyanato-4-methylbenzene
CETI-005	95808-48-3	hexadecyl p-tolylcarbamate
CETI-006	890655-07-9	hexadecyl (2-bromo-4-methylphenyl)carbamate
CETI-007	890655-08-0	2-(((hexadecyloxy)carbonyl)amino)-5-methylbenzoic acid

OptimisedRoute 3Steps 4 · Total yield 18.5 g

Synthetic routes & intermediates Route 3

Code	CAS No.	Intermediate
CETI-002	26272-90-2	hexadecyl carbonochloridate
CETI-003	2941-78-8	2-amino-5-methylbenzoic acid
CETI-007	890655-08-0	2-(((hexadecyloxy)carbonyl)amino)-5-methylbenzoic acid
CETI-008	1620769-74-5	methyl 2-amino-5-methylbenzoate sulfate
CETI-009	1620769-67-6	methyl 2-(((hexadecyloxy)carbonyl)amino)-5-methylbenzoate

Frequently asked questions

What are the approved indications of Cetilistat?

Approved indications include: 肥胖症.

When does the Cetilistat patent expire?

No public expiry year is available for Cetilistat yet; this page updates once verified.

How many synthesis routes are recorded for Cetilistat?

3 synthesis routes are recorded; the shortest is 2 steps with 2.51 g total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Cetilistat intermediates?

All intermediates in Cetilistat routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Cetilistat intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-24