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CAS 542-78-9

1,3-Propanedial

Codes: (II)115092-10-a

Application context (from source-drug indications)

GlaucomaProxodolol hydrochloride/Pilocarpine Hydrochloride闭角型青光眼Pilocarpine HydrochlorideOcular hypertensionPilocarpine HydrochlorideOpen-angle glaucomaPilocarpine Hydrochloride瞳孔缩小Pilocarpine HydrochlorideSjögren's syndromePilocarpine Hydrochloride虹膜炎Pilocarpine Hydrochloride

Source drugs (routes using this intermediate)

DrugTierExpiry
Proxodolol hydrochloride/Pilocarpine HydrochlorideTier C — Watch / trade-
Pilocarpine HydrochlorideTier C — Watch / trade-

Position in synthesis routes (up/downstream chain)

Ordered by route registration; left → right is the synthesis direction. The highlighted node is the current CAS; others link to their own profiles.

Proxodolol hydrochloride/Pilocarpine HydrochlorideOptimised routesteps: 6total yield: /
Methyl (2S)-2-hydroxybutanoate→1,3-Propanedial→Methyl (2S)-2-ethyl-3-formyl-4-oxobutanoate→Methyl (2S)-2-ethyl-4-hydroxy-3-(hydroxymethyl)butanoate→(3S)-3-Ethyl-4-(hydroxymethyl)oxolan-2-one→5-Chloro-1-methyl-1H-imidazole→(3S)-3-Ethyl-4-(1-methyl-1H-imidazole-5-carbonyl)oxolan-2-one→(3S)-3-Ethyl-4-[(1-methyl-1H-imidazol-5-yl)methyl]oxolan-2-one
Pilocarpine HydrochlorideOptimised routesteps: 6total yield: /
Methyl (2S)-2-hydroxybutanoate→1,3-Propanedial→Methyl (2S)-2-ethyl-3-formyl-4-oxobutanoate→Methyl (2S)-2-ethyl-4-hydroxy-3-(hydroxymethyl)butanoate→(3S)-3-Ethyl-4-(hydroxymethyl)oxolan-2-one→5-Chloro-1-methyl-1H-imidazole→(3S)-3-Ethyl-4-(1-methyl-1H-imidazole-5-carbonyl)oxolan-2-one→(3S)-3-Ethyl-4-[(1-methyl-1H-imidazol-5-yl)methyl]oxolan-2-one

Intermediates available on this site

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This is a CAS-level registry record: registrations across routes are merged. Supplier offers and buyer demands will be matched on this CAS as the primary key.