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Pharmaceutical Intermediates

Full official intermediate catalog + key intermediates with CEP / DMF / GMP / cold-chain qualifications and capacity details · each quotable via RFQ

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Orforglipron intermediates

样品订单(各 500g)+ 0.5KG 复购

2 deals completed · latest 2026-09-21

Documents in progress

Dealt

PINACOLONE

两用物项贸易品类

2 deals completed · latest 2026-01-19

Documents in progress

Dealt

4-(3-Bromophenyl)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline

CAS 543737-10-6

1 deal completed · latest 2026-07-08

Documents in progress

By Therapeutic Area of Target Drug

Click a class to filter both sections below; classes follow the target API's primary indication

Qualified Key IntermediatesCEP / DMF / GMP / Cold-chain / Capacity / Price-band details

13 items
Product / CASPurity / Impurity profile (redacted)Synthesis route (redacted)CapacityQualificationsPackaging / Cold-chainMOQ / Price bandAction
Lenacapavir INT-1|N-Boc 手性胺酯
CAS 1620056-47-4 · Antivirals
Target drug: lenacapavir
高保密
≥99.0%
单杂 ≤0.10%,总杂 ≤0.50%(脱敏)
手性还原 + Boc 保护(脱敏简述)1,200 kg/yr
US DMF
5 kg / 25 kg 桶(铝箔袋内衬)
1 kg
US$ 2,600-3,800 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-2|4-氯-7-硼酸酯吲唑
CAS 2189684-53-3 · Antivirals
Target drug: lenacapavir
高保密
≥98.5%
有关物质谱见 CDA 资料室
吲唑构建 + Miyaura 硼化(脱敏简述)900 kg/yr
US DMF
1 kg / 5 kg 铝瓶
Cold chain
0.5 kg
US$ 4,200-6,000 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-3|环丙烷并环戊烷吡唑乙酸
CAS 1620056-83-8 · Antivirals
Target drug: lenacapavir
高保密
≥99.0%
手性纯度 ≥99.5% ee(脱敏)
双环构建 + 三氟甲基化(脱敏简述)700 kg/yr
US DMF
1 kg 铝瓶
Cold chain
0.5 kg
US$ 5,800-8,200 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-4|3-甲基-3-(甲磺酰基)-1-丁炔
CAS 2109226-54-0 · Antivirals
Target drug: lenacapavir
CDA 后可看
≥98.0%
单杂 ≤0.20%(脱敏)
炔基化 + 砜基引入(脱敏简述)2,400 kg/yr
25 kg 桶
5 kg
US$ 780-1,150 / kg
Unibest Taizhou GMP-like Site
Lenacapavir (GS-6207) API
CAS 2189684-44-2 · Antivirals
Target drug: lenacapavir
高保密
≥99.5%
单杂 ≤0.10%,总杂 ≤0.30%(脱敏)
汇聚式偶联 + 成盐(脱敏简述)300 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶(密闭系统)
Cold chain
100 g
🔒 CDA 后开放
Unibest Nantong cGMP Site
Doravirine INT-1|3-氯-5-[(吡啶基)氧基]苯甲腈
CAS 1155846-86-8 · Antivirals
Target drug: doravirine
CDA 后可看
≥99.0%
单杂 ≤0.15%(脱敏)
芳香亲核取代成醚(脱敏简述)3,600 kg/yr
US DMFEU GMP
25 kg 桶
10 kg
US$ 420-620 / kg
Qualified Partner — East China API Works
Doravirine INT-2|3-氯-5-碘苯酚
CAS 861347-86-6 · Antivirals
Target drug: doravirine
≥99.0%
单杂 ≤0.15%(脱敏)
选择性碘代(脱敏简述)5,200 kg/yr
25 kg 桶
25 kg
US$ 210-320 / kg
Qualified Partner — East China API Works
Entecavir INT-1|嘌呤核苷中间体
CAS 142217-80-9 · Antivirals
Target drug: entecavir
≥99.0%
单杂 ≤0.10%(脱敏)
糖苷化 + 保护基策略(脱敏简述)1,800 kg/yr
CEPUS DMFEU GMP
5 kg / 25 kg 桶
5 kg
US$ 1,150-1,700 / kg
Qualified Partner — East China API Works
Belzutifan INT-1|(R)-3-氟-5-[(茚满酮基)氧基]苯甲腈
CAS 2738675-96-0 · Anti-cancer
Target drug: belzutifan
高保密
≥99.0%
手性纯度 ≥99.5% ee(脱敏)
手性还原 + 成醚(脱敏简述)800 kg/yr
US DMF
1 kg / 5 kg 铝瓶
1 kg
US$ 3,400-4,900 / kg
Unibest Taizhou GMP-like Site
Belzutifan INT-2|3-[(茚满酮基)氧基]-5-氟苯甲腈
CAS 1672665-55-2 · Anti-cancer
Target drug: belzutifan
高保密
≥99.0%
单杂 ≤0.10%(脱敏)
成醚 + 砜基氧化(脱敏简述)1,100 kg/yr
5 kg 桶
2 kg
US$ 2,100-3,100 / kg
Unibest Taizhou GMP-like Site
2'-dG(iBu) 亚磷酰胺单体
CAS 68892-42-2 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)400 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,600-2,400 / 100g
Unibest Nantong cGMP Site
2'-dA(Bz) 亚磷酰胺单体
CAS 4546-72-9 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)400 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,480-2,200 / 100g
Unibest Nantong cGMP Site
2'-dC(Bz) 亚磷酰胺单体
CAS 4836-13-9 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)350 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,520-2,280 / 100g
Unibest Nantong cGMP Site

Official Intermediate Full CatalogWith CAS numbers · Aggregated by target drug

Total 493 intermediates · covering 255 target drugs
Intermediate nameCAS No.Target drugAction
N-(4-cyanophenyl)-Glycine42288-26-6Dabigatran etexilate mesylate
2-chloro-4-methylpyrimidine13036-57-2Dabrafenib Mesylate
2,2,2-Trimethylthioacetamide630-22-8Dabrafenib Mesylate
2,6-Difluorobenzenesulfonyl chloride60230-36-6Dabrafenib Mesylate
Methyl 3-(2,6-difluorophenylsulfonaMido) -2-fluorobenzoate1195768-19-4Dabrafenib Mesylate
Methyl 3-amino-2-fluorobenzoate1195768-18-3Dabrafenib Mesylate
(2E)-4-(1-Piperidinyl)-2-butenoic acid hydrochloride197892-69-6Dacomitinib
(2S,4R)-1-(tert-butoxycarbonyl)-4-fluoropyrrolidine-2-carboxylic acid203866-14-2Danicopan
(2S,4R)-N-(6-bromopyridin-2-yl)-4-fluoropyrrolidine-2-carboxamide1903745-21-0Danicopan
1-(5-Bromo-1H-indazol-3-yl)ethan-1-one886363-74-2Danicopan
2-MethylpyriMidine-5-boronic Acid Pinacol Ester1052686-67-5Danicopan
(S)-2-Methylpyrrolidine-2- carboxylic acid hydrochloride1508261-86-6Daridorexant Hydrochloride
2-Methyl-L-proline Methyl ester hydrochloride220060-08-2Daridorexant Hydrochloride
4-Chloro-3-Methylbenzene-1,2- diaMine hydrochloride1087743-89-2Daridorexant Hydrochloride
5-methoxy-2-(2H-1,2,3-triazol-2- yl)benzoic acid1293284-55-5Daridorexant Hydrochloride
4-Bromo-2-chlorobenzonitrile154607-01-9Darolutamide
(E)-N-(2-Chloro-6-methylphenyl)-3-ethoxyacrylamide863127-76-8Dasatinib Hydrate
2-Amino-N-(2-chloro-6-methylphenyl)thiazole-5-carboxamide302964-24-5Dasatinib Hydrate
3,5-Difluoropyridine-2,6-diamine247069-27-8Delafloxacin meglumine
1,6-Diazaspiro[3.4]octane, 3-methyl-1-(phenylmethyl)-, ethanedioate (2:1), (3S,4R)-2230683-29-9Delgocitinib
6,7-Isoquinolinediol, 3,4-dihydro-hydrobromide (1:1)4593-96-8Deutetrabenazine
9,10-dihydroxy-3-isobutyl-3,4,6,7-tetrahydro-1H-pyrido[2,1-a]isoquinolin-2(11bH)-one89929-27-1Deutetrabenazine
Isoquinoline, 3,4-dihydro-6,7-di(methoxy-d3)-, hydrochloride (1:1)1783808-87-6Deutetrabenazine
1-Tritylimidazole-4-carboxaldehyde33016-47-6Dexmedetomidine Hydrochloride
(1S,4S,5S)-4-bromo-6-oxabicyclo[3.2.1]octan-7-one139893-81-5Edoxaban tosylate monohydrate
(S)-cyclohex-3-enecarboxylic acid5708-19-0Edoxaban tosylate monohydrate
2-[(5-Chloropyridin-2-yl)amino]-2-oxoacetic acid ethyl ester monohydrochloride1243308-37-3Edoxaban tosylate monohydrate
2-Bromo-5-methy1-4,5,6,7-tetrahydrothiazolo[5,4 -c]pyridine143150-92-9Edoxaban tosylate monohydrate
2-Bromo-5-methy1-4,5,6,7-tetrahydrothiazolo[5,4 -c]pyridine 4-methylbenzenesulfonate852291-42-0Edoxaban tosylate monohydrate
5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride720720-96-7Edoxaban tosylate monohydrate
Edoxaban tosylate monohydrate1229194-11-9Edoxaban tosylate monohydrate
N-(5-Chloropyridin-2-yl)oxalaMic acid ethyl ester349125-08-2Edoxaban tosylate monohydrate
tert-butyl (1R,2S,5S)-2-aMino-5-(diMethylcarbaMoyl)cyclohexylcarbaMate365998-36-3Edoxaban tosylate monohydrate
tert-Butyl [(1R,2S,5S)-2-amino-5-[(dimethylamino)carbonyl]cyclohexyl]carbamate oxalate1210348-34-7Edoxaban tosylate monohydrate
1-[2-fluoro-6-(trifluoromethyl)benzyl]-5-iodo-6-methylpyrimidine-2,4(1H,3H)-dione1150560-54-5Elagolix Sodium
1-[2-fluoro-6-(trifluoromethyl)benzyl]-6-methylpyrimidine-2,4(1H,3H)-dione830346-47-9Elagolix Sodium
5-(2-Fluoro-3-methoxyphenyl)-1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methyl-2,4(1H,3H)-pyrimidinedione1150560-59-0Elagolix Sodium
5-Bromo-1-(2-fluoro-6-trifluoromethyl-benzyl)-6- methyl-1H-pyrimidine-2,4-dione830346-48-0Elagolix Sodium
N-[(1R)-2-[(Methylsulfonyl)oxy]-1-phenylethyl]carbamic acid 1,1-dimethylethyl ester102089-75-8Elagolix Sodium
(R)-tert-butyl 2-(2-(benzyloxycarbonylaMino)-2-phenylacetaMido)acetate439088-73-0Elobixibat
(R)-α-[N-(t-butoxycarbonylmethyl) carbamoyl]benzylamine439088-74-1Elobixibat
1,5-Benzothiazepin-8-ol, 3,3-dibutyl-2,3,4,5-tetrahydro-7-(methylthio)-5-phenyl-, 1,1-dioxide439088-16-1Elobixibat
2-(Bromomethyl)-2-butylhexanoic acid100048-86-0Elobixibat
7-bromo-3,3-dibutyl-8-methoxy-2,3-dihydrobenzo[b][1,4]thiazepin-4(5H)-one439089-27-7Elobixibat
2-Trifluoromethyl-6-pyridinecarboxylic acid131747-42-7Enasidenib Mesylate
4-Amino-2-trifluoromethylpyridine147149-98-2 Enasidenib Mesylate
6-(6-(trifluoromethyl)pyridin-2-yl)-1,3,5-triazine-2,4(1H,3H)-dione1446507-38-5Enasidenib Mesylate
6-Trifluoromethyl-pyridine-2-carboxylic acid methyl ester155377-05-2Enasidenib Mesylate
1,3,5-Triazine-2,4(1H,3H)-dione, 3-(1,1-dimethylethyl)-6-(ethylthio)-1360105-53-8Ensitrelvir(S-217622)
3-(chloromethyl)-1-methyl-1H-1,2,4-Triazole hydrochloride135206-76-7Ensitrelvir(S-217622)
6-(Ethylthio)-1-(2,4,5-trifluorobenzyl)-1,3,5-triazine-2,4(1H,3H)-dione2771355-74-7Ensitrelvir(S-217622)
6-chloro-2-methyl-2H-indazol-5-amine1893125-36-4Ensitrelvir(S-217622)
S-ethylisothiourea hydrobromide1071-37-0Ensitrelvir(S-217622)
(2R, 3S.4S)-2, 3, 4-tris(benzyloxy)-4-((R)-4-((benzyloxy)meth yl)-2, 2-dimeth yl-1, 3- dioxolan-4-yl)-1-(4-methylDiDerazin-1-yl)butan-1-one1431329-07-5Ertugliflozin
2-((benzyloxy)(4-ethoxyphenyl)methyl)-4-bromo-1-chlorobenzene1298086-15-3Ertugliflozin
1H-Pyrrole-3-carboxylic acid, 4-methyl-5-[2-(trifluoromethyl)phenyl]-, ethyl ester1631030-76-6Esaxerenone
Oxcarbazepine28721-07-5Eslicarbazepine
Ethyl 2-(3-Formyl-4-hydroxyphenyl)-4-methylthiazole-5-carboxylate161798-01-2Febuxostat
Ethyl 2-(4-hydroxyphenyl)-4-methylthiazole-5-carboxylate161797-99-5Febuxostat
3-Fluorobenzenesulfonyl chloride701-27-9Fexuprazan HCl