盐酸奥达特罗
Tier C — Watch / tradeOlodaterol Hydrochloride
Targets：ADRB2
Brand：Striverdi Respimat
Indications (approved)：慢性阻塞性肺疾病、慢性支气管炎、气肿
Regional status
Synthetic routes & intermediates3 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| OLOD-001 | 490-78-8 | 1-(2,5-dihydroxyphenyl)ethanone |
| OLOD-002 | 100-39-0 | (bromomethyl)benzene |
| OLOD-003 | 30992-63-3 | 1-(5-(benzyloxy)-2-hydroxyphenyl)ethanone |
| OLOD-004 | 861841-94-3 | 1-(5-(benzyloxy)-2-hydroxy-3-nitrophenyl)ethanone |
| OLOD-005 | 861841-90-9 | 1-(3-amino-5-(benzyloxy)-2-hydroxyphenyl)ethanone |
| OLOD-006 | 79-04-9Available | 2-chloroacetyl chloride |
| OLOD-007 | 869478-09-1 | 8-acetyl-6-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-008 | 124955-27-7 | 6-(benzyloxy)-8-(2-ethoxy-2-hydroxyacetyl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-009 | 56490-94-9 | 1-(4-methoxyphenyl)-2-methylpropan-2-amine |
| OLOD-010 | 693273-06-2 | 6-(benzyloxy)-8-(1-hydroxy-2-((1-(4-methoxyphenyl)-2-methylpropan-2-yl)amino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one hydrochloride |
| OLOD-011 | 693273-18-6 | 6-hydroxy-8-(1-hydroxy-2-((1-(4-methoxyphenyl)-2-methylpropan-2-yl)amino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one hydrochloride |
| Code | CAS No. | Intermediate |
|---|---|---|
| OLOD-003 | 30992-63-3 | 1-(5-(benzyloxy)-2-hydroxyphenyl)ethanone |
| OLOD-004 | 861841-94-3 | 1-(5-(benzyloxy)-2-hydroxy-3-nitrophenyl)ethanone |
| OLOD-005 | 861841-90-9 | 1-(3-amino-5-(benzyloxy)-2-hydroxyphenyl)ethanone |
| OLOD-006 | 79-04-9Available | 2-chloroacetyl chloride |
| OLOD-007 | 869478-09-1 | 8-acetyl-6-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-009 | 56490-94-9 | 1-(4-methoxyphenyl)-2-methylpropan-2-amine |
| OLOD-012 | 869478-10-4 | 6-(benzyloxy)-8-(2-chloroacetyl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-013 | 869478-11-5 | (R)-6-(benzyloxy)-8-(2-chloro-1-hydroxyethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-014 | 869478-12-6 | (R)-6-(benzyloxy)-8-(oxiran-2-yl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-015 | 869478-13-7 | (R)-6-(benzyloxy)-8-(1-hydroxy-2-((1-(4-methoxyphenyl)-2-methylpropan-2-yl)amino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| Code | CAS No. | Intermediate |
|---|---|---|
| OLOD-001 | 490-78-8 | 1-(2,5-dihydroxyphenyl)ethanone |
| OLOD-002 | 100-39-0 | (bromomethyl)benzene |
| OLOD-003 | 30992-63-3 | 1-(5-(benzyloxy)-2-hydroxyphenyl)ethanone |
| OLOD-004 | 861841-94-3 | 1-(5-(benzyloxy)-2-hydroxy-3-nitrophenyl)ethanone |
| OLOD-005 | 861841-90-9 | 1-(3-amino-5-(benzyloxy)-2-hydroxyphenyl)ethanone |
| OLOD-006 | 79-04-9Available | 2-chloroacetyl chloride |
| OLOD-007 | 869478-09-1 | 8-acetyl-6-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-009 | 56490-94-9 | 1-(4-methoxyphenyl)-2-methylpropan-2-amine |
| OLOD-010 | 693273-06-2 | 6-(benzyloxy)-8-(1-hydroxy-2-((1-(4-methoxyphenyl)-2-methylpropan-2-yl)amino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one hydrochloride |
| OLOD-014 | 869478-12-6 | (R)-6-(benzyloxy)-8-(oxiran-2-yl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-016 | 926319-53-1 | 6-(benzyloxy)-8-(2-bromoacetyl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
| OLOD-017 | - | (R)-6-(benzyloxy)-8-(2-bromo-1-hydroxyethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
Frequently asked questions
What are the approved indications of Olodaterol Hydrochloride?
Approved indications include: 慢性阻塞性肺疾病, 慢性支气管炎, 气肿.
When does the Olodaterol Hydrochloride patent expire?
No public expiry year is available for Olodaterol Hydrochloride yet; this page updates once verified.
How many synthesis routes are recorded for Olodaterol Hydrochloride?
3 synthesis routes are recorded; the shortest is 8 steps with 4.50 g total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Olodaterol Hydrochloride intermediates?
1 intermediate CAS of Olodaterol Hydrochloride are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.
How do I get a quote for Olodaterol Hydrochloride intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-09-24