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Pharmaceutical Intermediates

Full official intermediate catalog + key intermediates with CEP / DMF / GMP / cold-chain qualifications and capacity details · each quotable via RFQ

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Orforglipron intermediates

样品订单(各 500g)+ 0.5KG 复购

2 deals completed · latest 2026-09-21

Documents in progress

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PINACOLONE

两用物项贸易品类

2 deals completed · latest 2026-01-19

Documents in progress

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4-(3-Bromophenyl)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline

CAS 543737-10-6

1 deal completed · latest 2026-07-08

Documents in progress

By Therapeutic Area of Target Drug

Click a class to filter both sections below; classes follow the target API's primary indication

Qualified Key IntermediatesCEP / DMF / GMP / Cold-chain / Capacity / Price-band details

13 items
Product / CASPurity / Impurity profile (redacted)Synthesis route (redacted)CapacityQualificationsPackaging / Cold-chainMOQ / Price bandAction
Lenacapavir INT-1|N-Boc 手性胺酯
CAS 1620056-47-4 · Antivirals
Target drug: lenacapavir
高保密
≥99.0%
单杂 ≤0.10%,总杂 ≤0.50%(脱敏)
手性还原 + Boc 保护(脱敏简述)1,200 kg/yr
US DMF
5 kg / 25 kg 桶(铝箔袋内衬)
1 kg
US$ 2,600-3,800 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-2|4-氯-7-硼酸酯吲唑
CAS 2189684-53-3 · Antivirals
Target drug: lenacapavir
高保密
≥98.5%
有关物质谱见 CDA 资料室
吲唑构建 + Miyaura 硼化(脱敏简述)900 kg/yr
US DMF
1 kg / 5 kg 铝瓶
Cold chain
0.5 kg
US$ 4,200-6,000 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-3|环丙烷并环戊烷吡唑乙酸
CAS 1620056-83-8 · Antivirals
Target drug: lenacapavir
高保密
≥99.0%
手性纯度 ≥99.5% ee(脱敏)
双环构建 + 三氟甲基化(脱敏简述)700 kg/yr
US DMF
1 kg 铝瓶
Cold chain
0.5 kg
US$ 5,800-8,200 / kg
Unibest Nantong cGMP Site
Lenacapavir INT-4|3-甲基-3-(甲磺酰基)-1-丁炔
CAS 2109226-54-0 · Antivirals
Target drug: lenacapavir
CDA 后可看
≥98.0%
单杂 ≤0.20%(脱敏)
炔基化 + 砜基引入(脱敏简述)2,400 kg/yr
25 kg 桶
5 kg
US$ 780-1,150 / kg
Unibest Taizhou GMP-like Site
Lenacapavir (GS-6207) API
CAS 2189684-44-2 · Antivirals
Target drug: lenacapavir
高保密
≥99.5%
单杂 ≤0.10%,总杂 ≤0.30%(脱敏)
汇聚式偶联 + 成盐(脱敏简述)300 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶(密闭系统)
Cold chain
100 g
🔒 CDA 后开放
Unibest Nantong cGMP Site
Doravirine INT-1|3-氯-5-[(吡啶基)氧基]苯甲腈
CAS 1155846-86-8 · Antivirals
Target drug: doravirine
CDA 后可看
≥99.0%
单杂 ≤0.15%(脱敏)
芳香亲核取代成醚(脱敏简述)3,600 kg/yr
US DMFEU GMP
25 kg 桶
10 kg
US$ 420-620 / kg
Qualified Partner — East China API Works
Doravirine INT-2|3-氯-5-碘苯酚
CAS 861347-86-6 · Antivirals
Target drug: doravirine
≥99.0%
单杂 ≤0.15%(脱敏)
选择性碘代(脱敏简述)5,200 kg/yr
25 kg 桶
25 kg
US$ 210-320 / kg
Qualified Partner — East China API Works
Entecavir INT-1|嘌呤核苷中间体
CAS 142217-80-9 · Antivirals
Target drug: entecavir
≥99.0%
单杂 ≤0.10%(脱敏)
糖苷化 + 保护基策略(脱敏简述)1,800 kg/yr
CEPUS DMFEU GMP
5 kg / 25 kg 桶
5 kg
US$ 1,150-1,700 / kg
Qualified Partner — East China API Works
Belzutifan INT-1|(R)-3-氟-5-[(茚满酮基)氧基]苯甲腈
CAS 2738675-96-0 · Anti-cancer
Target drug: belzutifan
高保密
≥99.0%
手性纯度 ≥99.5% ee(脱敏)
手性还原 + 成醚(脱敏简述)800 kg/yr
US DMF
1 kg / 5 kg 铝瓶
1 kg
US$ 3,400-4,900 / kg
Unibest Taizhou GMP-like Site
Belzutifan INT-2|3-[(茚满酮基)氧基]-5-氟苯甲腈
CAS 1672665-55-2 · Anti-cancer
Target drug: belzutifan
高保密
≥99.0%
单杂 ≤0.10%(脱敏)
成醚 + 砜基氧化(脱敏简述)1,100 kg/yr
5 kg 桶
2 kg
US$ 2,100-3,100 / kg
Unibest Taizhou GMP-like Site
2'-dG(iBu) 亚磷酰胺单体
CAS 68892-42-2 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)400 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,600-2,400 / 100g
Unibest Nantong cGMP Site
2'-dA(Bz) 亚磷酰胺单体
CAS 4546-72-9 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)400 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,480-2,200 / 100g
Unibest Nantong cGMP Site
2'-dC(Bz) 亚磷酰胺单体
CAS 4836-13-9 · Nucleic Acids
Target drug: oligonucleotide
≥99.0%
单杂 ≤0.10%(脱敏)
核苷保护 + 亚磷酰化(脱敏简述)350 kg/yr
US DMFEU GMP
100 g / 1 kg 铝瓶
Cold chain
100 g
US$ 1,520-2,280 / 100g
Unibest Nantong cGMP Site

Official Intermediate Full CatalogWith CAS numbers · Aggregated by target drug

Total 493 intermediates · covering 255 target drugs
Intermediate nameCAS No.Target drugAction
3-Chloro-4-[(pyridin-2-yl)methyloxy]aniline524955-09-7Neratinib/ Pyrotinib
6-amino-4-(3-chloro-4-(pyridin-2-ylmethoxy)phenylamino) -7- ethoxyquinoline-3-carbonitrile848139-78-6Neratinib/ Pyrotinib
Methyl 5-acetaMido-2-aMino-4-ethoxybenzoate1222172-49-7Neratinib/ Pyrotinib
N-(4-Chloro-3-cyano-7-ethoxy-6-quinolinyl)848133-76-6Neratinib/ Pyrotinib
3-(4-Methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)aniline641571-11-1Nilotinib
3-[(Aminoiminomethyl)amino] -4-methylbenzoic acid ethyl ester mononitrate641569-96-2Nilotinib
4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzoic acid641569-94-0Nilotinib
(3E)-2,3-Dihydro-3-(methoxyphenylmethylene) -2-oxo-1H-indole-6- carboxylic acid methyl ester1168150-46-6Nintedanib Esylate
2-Chloro-N-methyl-N-(4-nitrophenyl)acetamide2653-16-9Nintedanib Esylate
Methyl 2-oxoindole-6-carboxylate14192-26-8Nintedanib Esylate
N-(4-Aminophenyl)-N-methyl-2-(4-methylpiperazin -1-yl)acetamide262368-30-9Nintedanib Esylate
Trimethyl orthobenzoate707-07-3Nintedanib Esylate
(S)-tert-butyl 3-(4-aMinophenyl)piperidine-1-carboxylate1171197-20-8Niraparib
Methyl 3-formyl-2-nitrobenzoate138229-59-1Niraparib
Oxygen-fluorine acid82419-35-0Ofloxacin
1-(Cyclopropylcarbonyl)piperazine hydrochloride1021298-67-8Olaparib
2-fluoro-5-((4-oxo-3,4-dihydrophthalazin -1-yl)Methyl)benzoic acid763114-26-7Olaparib
2-Fluoro-5-[(3-oxo-1(3H)-isobenzofuranylidene)methyl]benzonitrile763114-25-6Olaparib
2-Fluoro-5-formylbenzonitrile218301-22-5Olaparib
3-oxo-1,3-dihydroisobenzofuran-1-ylphosphonic acid61260-15-9Olaparib
3-Methoxythiophene-2-carbaldehyde35134-07-7Oliceridine
OMadacycline (tosylate)1075240-43-5Omadacycline toslate
[3-(2-Chloro-pyrimidin-4-yl)-phenyl]-methanol859517-90-1Pacritinib
2-((allyloxy)Methyl)-1-(2-chl oroethoxy)-4-nitrob937273-31-9Pacritinib
2-(2-chloroethoxy)-5-nitrobenzaldehyde110837-53-1Pacritinib
3-(allyloxymethyl)-4-(2-(pyrrolidin-1-yl)ethoxy)benzenamine937273-33-1Pacritinib
4-(3-(allyloxymethyl)phenyl)-2-chloropyrimidine937273-29-5Pacritinib
5-Methyl-3,4-diphenylisoxazole37928-17-9Parecoxib sodium
BOC-3,4-DEHYDRO-PRO-OH51154-06-4Paxlovid
Boceprevir InterMediates565456-77-1Paxlovid
Methyl N-Boc-L-proline-3-ene74844-93-2Paxlovid
2,3-Dimethyl-2H-indazol-6-amine hydrochloride635702-60-2/1444731-72-0Pazopanib Hydrochloride
3-Amino-6-methylbenzenesulfonamide9/7/6973Pazopanib Hydrochloride
3-Methyl-6-nitroindazole6494-19-5Pazopanib Hydrochloride
N-(2-chloropyrimidin-4-yl)-N,2,3-trimethyl-2H-indazol-6-amine444731-75-3Pazopanib Hydrochloride
Methyl 4-chloro-1Hpyrrolo[2,3-b]pyridine-5-carboxylate951625-93-7Peficitinib Hydrobromide
Trans-4-Amino-1-hydroxyadamantane62058-03-1Peficitinib Hydrobromide
3-(4-methoxyphenoxy)propan-1-amine100841-00-7Pemafibrate
n-butyl (S)-2-trifluoromethanesulfonyl-oxybutanoate907192-60-3Pemafibrate
(1S,4R)-methyl 4-(Boc-amino)cyclopent-2-enecarboxylate168683-02-1Peramivir
(3aR,4R,6S,6aS)-4-(tert-butoxycarbonylaMino)-3- (pentan-3-yl)-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-6-carboxylic acid316173-28-1Peramivir
(3aR,4R,6S,6aS)-4-[[(1,1-DiMethylethoxy)carbonyl]aMino]-3-(1-ethylpropyl)-3a,5,6,6a-tetrahydro-4H-cyclopent[d]isoxazole-6-carboxylic Acid Methyl Ester229613-93-8Peramivir
4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]benzoic acid1571888-11-3Pirtobrutinib
methyl 4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]benzoate2182032-85-3Pirtobrutinib
N-(4-(2,2-dicyanoacetyl)benzyl)-5-fluoro-2- methoxybenzamide2819683-07-1Pirtobrutinib
N-[[4-(2,2-dicyano-1-methoxy-vinyl)phenyl]methyl]-5-fluoro-2-methoxy-benzamide2764851-04-7Pirtobrutinib
3-Amino-2,6-piperidinedione hydrochloride24666-56-6Pomalidomide/ Lenalidomide
3-Ethynylimidazolo[1,2 -b]pyridazine943320-61-4Ponatinib Hydrochloride
4-(4-Methylpiperazin-1-ylmethyl)-3-trifluoromethylaniline694499-26-8Ponatinib Hydrochloride
1-(3-Methoxypropyl)-4-piperidinamine179474-79-4Prucalopride
Methyl 4-(acetylaMino)-3-broMo-2-(2-broMoethoxy)-5-chlorobenzoate748788-39-8Prucalopride
(5-tert-butyl-isoxazol-3-yl)-carbaMic acid phenyl ester81479-48-3Quizartinib
3-Amino-5-tert-butylisoxazole55809-36-4Quizartinib
4-(2-Chloroethyl)morpholine hydrochloride3647-69-6Quizartinib
1,2,6,7-Tetrahydro-8H-indeno[5,4-b]furan-8-one196597-78-1Ramelteon
2,3-Dihydrobenzofuran496-16-2Ramelteon
Acetonitrile, (1,2,6,7-tetrahydro-8H-indeno[5,4-b]furan-8-ylidene)-, (2E)-196597-79-2Ramelteon
Despropionyl Ramelteon Hydrochloride196597-80-5Ramelteon
4-Amino-3-fluorophenol399-95-1Regorafenib
4-cyclopropyl-2-fluoro-N-(5-fluoro-2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)benzamide1787294-47-6Remibrutinib