Oxycodone Hydrochloride Hydrate
Tier C — Watch / tradeOxycodone Hydrochloride Hydrate
Targets：Opioid receptors
Brand：Oxygesic, OxiNorm, Oxycodone NT, Rexista Oxycodone XR, OxyContin, OxiFast, OROS-oxycodone, OXAYDO, Oxecta, Oxycodone DETERx, OxyContin Neo, Endone, OxyQD, Eubine, Roxicodone, Rexista, Acurox
Indications (approved)：Pain, 急性疼痛, Chronic pain
Regional status
Synthetic routes & intermediates2 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| OXYC-001 | 115-37-7 | (4R,7aR,12bS)-7,9-dimethoxy-3-methyl-2,3,4,7a-tetrahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline |
| OXYC-002 | 508-54-3 | (4R,4aS,7aR,12bS)-4a-hydroxy-9-methoxy-3-methyl-2,3,4,4a-tetrahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinolin-7(7aH)-one |
| Oxycodone | 76-42-6 | (4R,4aS,7aR,12bS)-4a-hydroxy-9-methoxy-3-methyl-2,3,4,4a,5,6-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinolin-7(7aH)-one |
| Code | CAS No. | Intermediate |
|---|---|---|
| OXYC-003 | 2973-58-2 | 2-bromo-3-hydroxy-4-methoxybenzaldehyde |
| OXYC-004 | 115961-42-7 | 2-bromo-4-methoxy-3-(methoxymethoxy)benzaldehyde |
| OXYC-005 | 1638678-28-0 | (2-bromo-4-methoxy-3-(methoxymethoxy)phenyl)methanol |
| OXYC-006 | 1638678-29-1 | 2-bromo-1-(bromomethyl)-4-methoxy-3-(methoxymethoxy)benzene |
| OXYC-007 | 1638678-30-4 | (R)-4-benzyl-3-(2-(4-(benzyloxy)phenyl)acetyl)oxazolidin-2-one |
| OXYC-008 | - | (R)-4-benzyl-3-((R)-2-(4-(benzyloxy)-2-bromophenyl)-3-(4-methoxy-3-(methoxymethoxy)phenyl)propanoyl)oxazolidin-2-one |
| OXYC-009 | - | (R)-2-(4-(benzyloxy)-2-bromophenyl)-3-(4-methoxy-3-(methoxymethoxy)phenyl)propanoic acid |
| OXYC-010 | - | methyl (R)-2-(4-(benzyloxy)-2-bromophenyl)-3-(4-methoxy-3-(methoxymethoxy)phenyl)propanoate |
| OXYC-011 | 1638678-34-8 | methyl (R)-6-(benzyloxy)-3-methoxy-4-(methoxymethoxy)-9,10-dihydrophenanthrene-9-carboxylate |
| OXYC-012 | 1638678-38-2 | (R)-(6-hydroxy-3-methoxy-4-(methoxymethoxy)-9,10-dihydrophenanthren-9-yl)methyl acetate |
| OXYC-013 | 1638678-40-6 | ((8aR,9S)-8a-hydroxy-3-methoxy-4-(methoxymethoxy)-6-oxo-6,8a,9,10-tetrahydrophenanthren-9-yl)methyl acetate |
| OXYC-014 | 1638678-42-8 | ((8aR,9S)-8a-hydroxy-3-methoxy-4-(methoxymethoxy)-6-oxo-6,7,8,8a,9,10-hexahydrophenanthren-9-yl)methyl acetate |
| OXYC-015 | 37517-81-0 | methyl 3-chloro-3-oxopropanoate |
| OXYC-016 | 1638678-43-9 | (8aR,9S)-9-(acetoxymethyl)-3-methoxy-4-(methoxymethoxy)-6-oxo-7,8,9,10-tetrahydrophenanthren-8a(6H)-yl methyl malonate |
| OXYC-017 | - | methyl (4bS,8aR,9S,13S)-9-(acetoxymethyl)-3-methoxy-4-(methoxymethoxy)-6,12-dioxo-5,6,7,8,9,10-hexahydro-8a,4b-(epoxyethano)phenanthrene-13-carboxylate |
| OXYC-018 | 1638678-46-2 | ((4bS,8aR,9S)-3-methoxy-4-(methoxymethoxy)-6,12-dioxo-5,6,7,8,9,10-hexahydro-8a,4b-(epoxyethano)phenanthren-9-yl)methyl acetate |
| OXYC-019 | 1638678-47-3 | ((4bS,8aR,9S)-4-hydroxy-3-methoxy-6,12-dioxo-5,6,7,8,9,10-hexahydro-8a,4b-(epoxyethano)phenanthren-9-yl)methyl acetate |
| OXYC-020 | - | ((4bR,8aR,9S)-5-bromo-4-hydroxy-3-methoxy-6,12-dioxo-5,6,7,8,9,10-hexahydro-8a,4b-(epoxyethano)phenanthren-9-yl)methyl acetate |
| OXYC-021 | 1638678-50-8 | 7a,9c-(Epoxyethano)phenanthro[4,5-bcd]furan-5,11(4aH)-dione, 8-[(acetyloxy)methyl]-6,7,8,9-tetrahydro-3-methoxy-, (4aR,7aR,8S,9cS)- |
| OXYC-022 | 1638678-51-9 | 7a,9c-(Epoxyethano)phenanthro[4,5-bcd]furan-5,11(4aH)-dione, 6,7,8,9-tetrahydro-8-(hydroxymethyl)-3-methoxy-, (4aR,7aR,8S,9cS)- |
| OXYC-023 | 1638678-52-0 | 7a,9c-(Epoxyethano)phenanthro[4,5-bcd]furan-8-carboxylic acid, 4a,5,6,7,8,9-hexahydro-3-methoxy-5,11-dioxo-, (4aR,7aR,8R,9cS)- |
| OXYC-024 | 1638678-53-1 | 7a,9c-(Epoxyethano)phenanthro[4,5-bcd]furan-8-carboxamide, 4a,5,6,7,8,9-hexahydro-3-methoxy-5,11-dioxo-, (4aR,7aR,8R,9cS)- |
| OXYC-025 | 1638678-54-2 | (4R,4aS,7aR,12bS)-4a-hydroxy-9-methoxy-4,4a,5,6-tetrahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-2,7(3H,7aH)-dione |
| OXYC-026 | - | (4R,4aS,7aR,12bS)-9-methoxy-3-methyl-1,2,3,4,5,6,7,7a-octahydro-4aH-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,7-diol |
Frequently asked questions
What are the approved indications of Oxycodone Hydrochloride Hydrate?
Approved indications include: Pain, 急性疼痛, Chronic pain.
When does the Oxycodone Hydrochloride Hydrate patent expire?
No public expiry year is available for Oxycodone Hydrochloride Hydrate yet; this page updates once verified.
How many synthesis routes are recorded for Oxycodone Hydrochloride Hydrate?
2 synthesis routes are recorded; the shortest is 2 steps with 1.51 g (Oxycodone) total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Oxycodone Hydrochloride Hydrate intermediates?
All intermediates in Oxycodone Hydrochloride Hydrate routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.
How do I get a quote for Oxycodone Hydrochloride Hydrate intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-09-27